SCHEMBL4638511

SCHEMBL4638511

CC(C)(C)[Si](C)(C)OCCC#CC(O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1Cl

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637942 0.91 AKR1C3 (0.32) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4638484 0.81 AKR1C3 (0.35) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4638086 0.76 TACR1 (0.39) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4639492 0.76 HSP90AA1 (0.32) HSP90AA1HSP90AB1
SCHEMBL4637992 0.73 GRM2 (0.37) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4708145 0.73 AKR1C3 (0.36) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4639425 0.69 USP2 (0.35) AKR1C3HSP90AA1HSP90AB1
SCHEMBL18255823 0.66 IDO1 (0.33)
SCHEMBL4638930 0.65 ALDH1A1 (0.38) AKR1C3HSP90AA1HSP90AB1
SCHEMBL4706583 0.65 HTT (0.36) AKR1C3HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed