SCHEMBL4706583

SCHEMBL4706583

ON=Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ENPP2 Q13822 1/20 0.35
AKR1C3 P42330 2/20 0.35
GRM2 Q14416 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
PTGER4 P35408 4/20 0.33
POLB P06746 1/20 0.33
CASP1 P29466 1/20 0.33
CASP5 P51878 1/20 0.33
AKR1C2 P52895 1/20 0.32
PDE8B O95263 1/20 0.32
TSHR P16473 1/20 0.31
MAPT P10636 2/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638624 0.83 HSP90AA1 (0.38) HTTL3MBTL1ENPP2AKR1C3GRM2
SCHEMBL4705254 0.80 ALDH1A1 (0.41) HTTL3MBTL1AKR1C3GRM2HSP90AA1
SCHEMBL4708361 0.79 USP2 (0.37) HTTL3MBTL1AKR1C3GRM2HSP90AA1
SCHEMBL4708366 0.77 CASP1 (0.35) CASP1CASP5MAPTLMNANPSR1
SCHEMBL4707339 0.76 POLB (0.39) HTTL3MBTL1POLB
SCHEMBL4637929 0.74 HPGD (0.45) HTTL3MBTL1ENPP2AKR1C3JUN
SCHEMBL4759169 0.72 HTT (0.38) HTTL3MBTL1ENPP2AKR1C3GRM2
SCHEMBL4638906 0.68 CYP19A1 (0.49) AKR1C3MAPTTP53LMNANPSR1
SCHEMBL27603337 0.68 GRM2 (0.36) HTTL3MBTL1GRM2JUNNFKB1
SCHEMBL27603235 0.68 GRM2 (0.36) HTTL3MBTL1AKR1C3GRM2AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed