SCHEMBL4638554

SCHEMBL4638554

Cc1c(C(=O)C#Cc2ccccc2Cl)nnn1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
AKR1C3 P42330 2/20 0.38
TP53 P04637 2/20 0.38
GRM5 P41594 1/20 0.38
AKR1C2 P52895 1/20 0.38
MAPT P10636 4/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TACR1 P25103 1/20 0.36
CYP2C9 P11712 1/20 0.36
KLKB1 P03952 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637988 0.91 PTGDR2 (0.40) CCR1PTGDR2AKR1C3TP53GRM5
SCHEMBL4638053 0.87 ALDH1A1 (0.44) PTGDR2AKR1C3AKR1C2MAPTHTT
SCHEMBL4637813 0.84 IDH1 (0.39) PTGDR2AKR1C3AKR1C2SMN1; SMN2HTT
SCHEMBL4637949 0.84 IDH1 (0.39) PTGDR2AKR1C3TP53AKR1C2MAPT
SCHEMBL4707915 0.82 IDH1 (0.48) PTGDR2HTTL3MBTL1GAAALDH1A1
SCHEMBL4637887 0.82 USP2 (0.36) PTGDR2AKR1C3AKR1C2MEN1KMT2A
SCHEMBL4638552 0.81 TACR1 (0.40) CCR1PTGDR2AKR1C3AKR1C2MAPT
SCHEMBL4637824 0.76 ALDH1A1 (0.44) PTGDR2AKR1C3AKR1C2SMN1; SMN2GAA
SCHEMBL4637753 0.76 IDH1 (0.47) PTGDR2AKR1C3TP53AKR1C2MAPT
SCHEMBL4637729 0.76 PTGDR2 (0.41) PTGDR2SMN1; SMN2HTTGAATACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed