SCHEMBL4639698

SCHEMBL4639698

CCCCN1c2[nH]c(=O)[nH]c(=O)c2NC1c1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.36
ADORA2B P29275 8/20 0.33
ADORA1 P30542 5/20 0.33
ADORA2A P29274 4/20 0.33
ADORA3 P0DMS8 3/20 0.33
PDE9A O76083 2/20 0.33
PDE1C Q14123 1/20 0.33
PDE4A P27815 1/20 0.31
PREP P48147 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1697136 0.82 ADORA2B (0.47) ADORA2BADORA1ADORA2AADORA3
SCHEMBL5685834 0.72 ADORA2B (0.45) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4639695 0.72 ADORA2B (0.45) ADORA2BADORA1ADORA2AADORA3
SCHEMBL244428 0.65 ADORA2B (0.74) ADORA2BADORA1ADORA2AADORA3
SCHEMBL21491519 0.63 GLS (0.38) DAOADORA1ADORA3GRIN1GRIN2B
SCHEMBL26202009 0.62 CYP3A4 (0.40) DAOGRIN1GRIN2B
SCHEMBL30744539 0.62 PPARD (0.42) PREP
SCHEMBL21493002 0.62 PPARD (0.42) PREP
SCHEMBL25269987 0.62 GRIN1 (0.40) DAOGRIN1GRIN2B
SCHEMBL2684038 0.62 ADORA2B (0.54) ADORA2BADORA1ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622908-B1 XANTHINE DERIVATIVES AS A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-08-06 EP claimed