SCHEMBL4639740

SCHEMBL4639740

Clc1ccc(Oc2ccc(CSCc3ccc(Oc4ccc(Cl)cc4)cc3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP2C9 P11712 1/20 0.52
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP2D6 P10635 2/20 0.46
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
RAB9A P51151 1/20 0.45
IDO1 P14902 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
S1PR5 Q9H228 1/20 0.42
PPARG P37231 3/20 0.41
PPARA Q07869 3/20 0.41
GFER P55789 1/20 0.41
APP P05067 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3674399 0.86 CYP1A2 (0.63) CYP1A2CYP2C19CYP2C9ALDH1A1LMNA
SCHEMBL10870044 0.79 MAOB (0.56) MAOAMAOBIDO1S1PR5PPARG
SCHEMBL9242729 0.78 MAOA (0.74) CYP1A2CYP2C19CYP2C9MAOAMAOB
SCHEMBL457634 0.78 MAOA (0.74) CYP1A2CYP2C19CYP2C9MAOAMAOB
SCHEMBL10614200 0.77 TDP1 (0.56) CYP1A2CYP2C19CYP2C9ALDH1A1LMNA
SCHEMBL2987196 0.77 MAOB (0.54) MAOAMAOBIDO1S1PR5PPARG
SCHEMBL6446133 0.77 MAOB (0.48) MAOAMAOBALDH1A1LMNAS1PR5
SCHEMBL29738633 0.77 CYP1A2 (0.53) CYP1A2CYP2C19CYP2C9ALDH1A1LMNA
SCHEMBL4639745 0.76 IDO1 (0.73) MAOAMAOBIDO1S1PR5PPARG
SCHEMBL2056280 0.76 MAOB (0.52) CYP2C19MAOAMAOBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1240208-A Process for preparing 3-arylsulfur hydroxamic acids HOFFMANN LA ROCHE (CH) 2000-01-05 CN claimed
EP-1357109-B1 Process for aryl alkyl sulfide HOFFMANN LA ROCHE (CH) 2008-07-23 EP disclosed
EP-1357109-A2 Process for aryl alkyl sulfide F. HOFFMANN-LA ROCHE AG (CH) 2003-10-29 EP disclosed
CN-1388117-A Process for prodcing 3-aryl sulfate iso-hydroximic acid HOFFMANN LA ROCHE (CH) 2003-01-01 CN disclosed
CN-1240208-A Process for preparing 3-arylsulfur hydroxamic acids HOFFMANN LA ROCHE (CH) 2000-01-05 CN disclosed
EP-0965592-A1 Process for preparing 3-arylsulfur hydroxamic acids F. HOFFMANN-LA ROCHE AG (CH) 1999-12-22 EP disclosed