SCHEMBL4640337

SCHEMBL4640337

NC(=O)c1ccc(OBOc2ccc(C(N)=O)c(Cl)c2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
ATM Q13315 1/20 0.41
CHEK2 O96017 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
ADRA1D P25100 1/20 0.38
RAB9A P51151 5/20 0.37
MAPT P10636 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14484639 0.86 ALDH1A1 (0.45) KMT2AATMCHEK2CA12CA1
SCHEMBL29966096 0.80 KDM4E (0.54) KMT2ACA1CA2RAB9AMAPT
SCHEMBL2468448 0.80 KDM4E (0.54) KMT2ACA1CA2RAB9AMAPT
SCHEMBL516293 0.79 ABL1 (0.46) KMT2AATMCA12CA1CA2
SCHEMBL4640347 0.78 JAK2 (0.46) KMT2ARAB9AMAPTSMN1; SMN2NPC1
SCHEMBL2104774 0.77 PARP10 (0.56) KMT2AMKNK1MKNK2CA12CA1
SCHEMBL9901975 0.76 AKR1C2 (0.47) KMT2AMKNK1MKNK2KDM4EJAK2
SCHEMBL28039268 0.76 PARP10 (0.56) KMT2AATMCHEK2ALDH1A1
SCHEMBL15544328 0.75 DGAT1 (0.41) KMT2AMAPTCASP1ALDH1A1
SCHEMBL4687865 0.75 SMN1; SMN2 (0.44) KMT2AMKNK1MKNK2CHEK2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964834-A1 Sulphonyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-09-03 EP disclosed
EP-1956016-A1 Bicyclic acyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-08-13 EP disclosed