SCHEMBL4640764

SCHEMBL4640764

O=C(O)c1cnccc1CCN1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
SLC6A3 Q01959 1/20 0.40
KDM4C Q9H3R0 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KDM6B O15054 1/20 0.39
KDM4A O75164 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
KDM4D Q6B0I6 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
CACNA1B Q00975 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6035089 0.79 HRH3 (0.45) HRH3L3MBTL1TDP1CYP1A2CYP3A4
SCHEMBL9858541 0.76 KDM4C (0.47) L3MBTL1TDP1KDM4CALDH1A1KMT2A
SCHEMBL6034963 0.75 HRH3 (0.54) HRH3L3MBTL1TDP1CYP1A2CYP3A4
SCHEMBL28079169 0.74 KDM4C (0.46) L3MBTL1TDP1KDM4CALDH1A1KMT2A
SCHEMBL11284708 0.74 FOLH1 (0.58) L3MBTL1TDP1KDM4CALDH1A1KMT2A
SCHEMBL258369 0.74 KDM4C (0.51) L3MBTL1TDP1CYP1A2CYP3A4KDM4C
SCHEMBL169608 0.74 KDM4E (0.38) TDP1CYP3A4KDM4CALDH1A1KMT2A
Hydrochloric Acid SCHEMBL5739434 0.73 KDM4C (0.50) L3MBTL1TDP1CYP1A2CYP3A4KDM4C
SCHEMBL123203 0.72 KDM4C (0.51) L3MBTL1TDP1KDM4CALDH1A1KMT2A
SCHEMBL3880004 0.72 KDM4C (0.50) L3MBTL1TDP1KDM4CALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885697-A2 SOLUBLE EPOXIDE HYDROLASE INHIBITORS AND METHODS OF USING SAME BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-02-13 EP disclosed
WO-2006121719-A2 SOLUBLE EPOXIDE HYDROLASE INHIBITORS AND METHODS OF USING SAME BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2006-11-16 WO disclosed