SCHEMBL4644396

SCHEMBL4644396

NCC1(N2CCCC(COCc3ccccc3)C2)CCC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
CTSK P43235 1/20 0.48
CHRNB2 P17787 2/20 0.41
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
NAAA Q02083 1/20 0.38
TAAR1 Q96RJ0 1/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3058053 0.78 CTSL (0.43) CTSLCTSBCTSKNAAATAAR1
SCHEMBL27685353 0.73 CTSK (0.56) CTSLCTSBCTSKCHRNB2CHRNB4
SCHEMBL22616971 0.71 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNB4
SCHEMBL22616969 0.71 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNB4
SCHEMBL22616980 0.71 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNB4
SCHEMBL6649338 0.71 TSHR (0.54) CTSLCTSBCTSKNAAATAAR1
SCHEMBL4677170 0.71 TSHR (0.54) CTSLCTSBCTSKNAAATAAR1
SCHEMBL1700657 0.70 CTSL (0.45) CTSLCTSBCTSKNAAATAAR1
SCHEMBL2701945 0.70 CTSL (0.53) CTSLCTSBCTSKNAAATAAR1
Hydrochloric Acid SCHEMBL5516807 0.69 CTSL (0.44) CTSLCTSBCTSKNAAATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960360-A1 AZETIDINE DERIVATIVES AS GLYT1 INHIBITORS MERCK SHARP & DOHME LTD. (GB) 2008-08-27 EP disclosed
WO-2007060484-A1 AZETIDINE DERIVATIVES AS GLYT1 INHIBITORS MERCK SHARP & DOHME LIMITED (GB) 2007-05-31 WO disclosed