SCHEMBL464457

SCHEMBL464457

COC(=O)SSCCNC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
IDO1 P14902 3/20 0.44
EPHX1 P07099 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GFER P55789 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1082707 0.86 TDP1 (0.56) TDP1MEN1KMT2AGAAIDO1
SCHEMBL25014915 0.79 TDP1 (0.50) TDP1MEN1KMT2AGAAIDO1
SCHEMBL10037268 0.79 TDP1 (0.50) TDP1MEN1KMT2AGAAIDO1
SCHEMBL15083132 0.79 TDP1 (0.50) TDP1MEN1KMT2AGAAIDO1
SCHEMBL1042383 0.79 TDP1 (0.59) TDP1MEN1KMT2AGAAIDO1
SCHEMBL14646688 0.79 TDP1 (0.50) TDP1MEN1KMT2AGAAIDO1
SCHEMBL12103908 0.78 TDP1 (0.49) TDP1MEN1KMT2AGAAIDO1
SCHEMBL1584489 0.78 TDP1 (0.49) TDP1MEN1KMT2AGAAIDO1
SCHEMBL14755649 0.78 TDP1 (0.49) TDP1MEN1KMT2AGAAIDO1
SCHEMBL903325 0.78 TDP1 (0.49) TDP1MEN1KMT2AGAAIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250057960-A1 OLIGOSACCHARIDE COMPLEXES AND USES BioNTech SE (DE) 2025-02-20 US disclosed
US-20250002522-A1 OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2025-01-02 US disclosed
US-20240417418-A1 DISULFIDE OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2024-12-19 US disclosed
EP-4401788-A1 OLIGOSACCHARIDE COMPLEXES AND USES BioNTech SE (DE) 2024-07-24 EP disclosed
EP-4402149-A1 DISULFIDE OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2024-07-24 EP disclosed
EP-4402150-A1 OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2024-07-24 EP disclosed
EP-4286394-A1 OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2023-12-06 EP disclosed
EP-4286004-A1 DISULFIDE OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2023-12-06 EP disclosed
WO-2023067126-A1 OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2023-04-27 WO disclosed
WO-2023067124-A1 DISULFIDE OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES BioNTech SE (DE) 2023-04-27 WO disclosed
US-20200046845-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CERULEAN PHARMA INC. 2020-02-13 US disclosed
EP-3566719-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASES Cerulean Pharma Inc. (US) 2019-11-13 EP disclosed
US-20180193486-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE CERULEAN PHARMA INC. 2018-07-12 US disclosed
US-20160058874-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CERULEAN PHARMA INC. (US) 2016-03-03 US disclosed
US-20150005230-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CERULEAN PHARMA INC. (US) 2015-01-01 US disclosed
US-20140255374-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE CERULEAN PHARMA INC. (US) 2014-09-11 US disclosed
WO-2013116200-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CERULEAN PHARMA INC. (US) 2013-08-08 WO disclosed
US-20130196906-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CERULEAN PHARMA INC. (US) 2013-08-01 US disclosed
US-20120064107-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE CERULEAN PHARMA INC. (US) 2012-03-15 US disclosed
WO-2011146638-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASES CERULEAN PHARMA INC. (US) 2011-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180193486-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE PHOSPHO1, SGMS1, SGMS2 TDP1 1801/4885MEN1 1397/4885KMT2A 3696/4885
US-20250057960-A1 OLIGOSACCHARIDE COMPLEXES AND USES CD4, FUT6, UGCG TDP1 4398/4885MEN1 3067/4885KMT2A 4793/4885
US-20130196906-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CDR2, DDOST, GALC TDP1 1095/4885MEN1 2879/4885KMT2A 4529/4885
US-20250002522-A1 OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES OSTC, FUT6, MAN2B2 TDP1 1306/4885MEN1 2389/4885KMT2A 4165/4885
US-20140255374-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE PHOSPHO1, SGMS1, SGMS2 TDP1 1801/4885MEN1 1397/4885KMT2A 3696/4885
US-20120064107-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF AUTOIMMUNE AND OTHER DISEASE PHOSPHO1, SGMS1, SGMS2 TDP1 1801/4885MEN1 1397/4885KMT2A 3696/4885
US-20200046845-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CDR2, DDOST, GALC TDP1 1095/4885MEN1 2879/4885KMT2A 4529/4885
US-20240417418-A1 DISULFIDE OLIGOSACCHARIDE COMPOUNDS AND COMPLEXES DNAJC10, SNRPA, SNRPA1 TDP1 2292/4885MEN1 3682/4885KMT2A 4190/4885
US-20150005230-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CDR2, DDOST, GALC TDP1 1095/4885MEN1 2879/4885KMT2A 4529/4885
US-20160058874-A1 CYCLODEXTRIN-BASED POLYMERS FOR THERAPEUTIC DELIVERY CDR2, DDOST, GALC TDP1 1095/4885MEN1 2879/4885KMT2A 4529/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.