SCHEMBL4645453

SCHEMBL4645453

CCOC(=O)Oc1ccc2ncn(CCC(C)(C)NCC(O)c3cccc(NS(=O)(=O)c4ccccc4)c3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 12/20 0.45
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
HPGD P15428 2/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
ADRA1A P35348 3/20 0.36
NR1I2 O75469 1/20 0.36
ALDH1A1 P00352 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640763 1.00 ADRB3 (0.45) ADRB3OPRM1OPRD1HPGDMTNR1A
SCHEMBL4640303 0.94 ADRB3 (0.47) ADRB3OPRM1OPRD1HPGDADRA1A
SCHEMBL4643457 0.94 ADRB3 (0.47) ADRB3OPRM1OPRD1HPGDADRA1A
SCHEMBL4840747 0.90 ADRB3 (0.42) ADRB3OPRM1OPRD1HPGDNR1I2
Trifluoroacetic Acid SCHEMBL4644103 0.89 ADRB3 (0.45) ADRB3OPRM1OPRD1HPGDADRA1A
SCHEMBL5468010 0.89 ADRB3 (0.43) ADRB3OPRM1OPRD1HPGDALDH1A1
SCHEMBL4913365 0.89 ADRB3 (0.43) ADRB3OPRM1OPRD1HPGDALDH1A1
SCHEMBL4776666 0.88 ADRB3 (0.42) ADRB3OPRM1OPRD1HPGDNR1I2
SCHEMBL4777081 0.88 ADRB3 (0.42) ADRB3OPRM1OPRD1HPGDNR1I2
SCHEMBL4775581 0.87 ADRB3 (0.42) ADRB3OPRM1OPRD1HPGDNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed