SCHEMBL4649199

SCHEMBL4649199

COc1ccc(Cc2cc(F)c3c(=O)c(C(=O)O)c[nH]c3c2F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 3/20 0.39
HTT P42858 3/20 0.39
MAPK1 P28482 2/20 0.39
RAB9A P51151 1/20 0.39
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
SLC5A2 P31639 1/20 0.38
GSK3B P49841 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALKBH1 Q13686 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650790 0.87 KDM5A (0.42) ALDH1A1HPGDKDM4EHTTCSNK2A2
SCHEMBL4650011 0.86 KDM4C (0.45) ALDH1A1HPGDKDM4ERAB9ACSNK2A2
SCHEMBL4650143 0.84 CSNK2A2 (0.43) ALDH1A1HPGDKDM4ELMNACSNK2A2
SCHEMBL4559012 0.81 CHRM1 (0.43) ALDH1A1HPGDCSNK2A2CSNK2BCSNK2A1
SCHEMBL4650001 0.80 CSNK2A2 (0.39) ALDH1A1HPGDCSNK2A2CSNK2BCSNK2A1
SCHEMBL4649448 0.80 CSNK2A1 (0.44) ALDH1A1HPGDKDM4ELMNACSNK2A2
SCHEMBL4650109 0.80 CYP1A2 (0.46) ALDH1A1HPGDKDM4EHTTCSNK2A2
SCHEMBL4650040 0.78 KDM4E (0.46) ALDH1A1HPGDKDM4ELMNAHTT
SCHEMBL4650643 0.78 KDM5A (0.41) ALDH1A1HPGDCSNK2A2CSNK2BCSNK2A1
SCHEMBL1126554 0.78 CSNK2A2 (0.38) ALDH1A1HPGDKDM4ECSNK2A2CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed