SCHEMBL4649685

SCHEMBL4649685

CCOCCc1cc(C(=O)Cl)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
EPHX2 P34913 1/20 0.33
TSHR P16473 2/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 3/20 0.32
DAO P14920 3/20 0.31
P2RX7 Q99572 1/20 0.31
HCRTR1 O43613 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
BAZ2A Q9UIF9 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649373 0.87 NOTUM (0.42) KMT2ATDP1MEN1POLBEPHX2
SCHEMBL4649821 0.85 ALDH1A1 (0.34) EPHX2ALDH1A1DAOHCRTR1BAZ2B
SCHEMBL4649101 0.81 GRIN2D (0.35) EPHX2ALDH1A1DAOHCRTR1BAZ2B
SCHEMBL4648846 0.72 NOTUM (0.44) TDP1EPHX2ALDH1A1DAOBAZ2B
SCHEMBL27748064 0.70 CYP4F2 (0.43) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL6207336 0.69 NOTUM (0.48) KMT2ATDP1EPHX2ALDH1A1
SCHEMBL22623624 0.68 CA12 (0.47) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL27704327 0.68 TPMT (0.38) KMT2ATDP1MEN1POLBTSHR
SCHEMBL8061456 0.67 PLK1 (0.40) POLBTSHRALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL6209517 0.66 NOTUM (0.53) KMT2ATDP1MEN1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960367-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2008-08-27 EP disclosed
WO-2007067836-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-06-14 WO disclosed