SCHEMBL4654947

SCHEMBL4654947

CCOC(=O)C1=CCNC=C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
MAPT P10636 3/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.39
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA7 P43166 3/20 0.37
CA9 Q16790 3/20 0.37
CA14 Q9ULX7 3/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
CYP1A2 P05177 3/20 0.36
LMNA P02545 3/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19434085 0.77 THRB (0.41) TSHRCA1CA2ALDH1A1POLB
SCHEMBL13969442 0.73 TSHR (0.42) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL5552082 0.72 TSHR (0.39) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL27630535 0.72 KMT2A (0.40) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL5114658 0.71 CA12 (0.43) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL4467924 0.71 ALDH1A1 (0.41) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL47924 0.70 CA12 (0.42) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL1180315 0.70 KDM4E (0.38) KDM4EKMT2AMEN1MAPTALOX15
SCHEMBL16229717 0.69
SCHEMBL28381747 0.69 TSHR (0.39) KDM4EKMT2AMEN1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116942663-A Compounds for the treatment of HBV 葛兰素史克知识产权开发有限公司 2023-10-27 CN disclosed
EP-1996588-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS Torrent Pharmaceuticals Ltd (IN) 2008-12-03 EP disclosed
WO-2007100295-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS TORRENT PHARMACEUTICALS LTD (IN) 2007-09-07 WO disclosed