SCHEMBL4655293

SCHEMBL4655293

Cn1ccc2cc(NC(=O)c3cc4cc(F)ccc4n3Cc3ccc(C(C)(C)C)cc3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 11/20 0.46
EPHX2 P34913 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
PPARG P37231 1/20 0.45
CCR9 P51686 3/20 0.44
CCR2 P41597 1/20 0.44
MAPT P10636 2/20 0.44
KCNQ3 O43525 1/20 0.44
KCNQ2 O43526 1/20 0.44
KCNQ4 P56696 1/20 0.44
KCNQ5 Q9NR82 1/20 0.44
TP53 P04637 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4655354 0.93 KCNQ3 (0.50) ECE1PPARGCCR2MAPTKCNQ3
SCHEMBL4656519 0.92 ECE1 (0.54) ECE1EPHX2NR1H4
SCHEMBL4655328 0.89 PTGS2 (0.46) ECE1CCR2MAPTTP53KDM4E
SCHEMBL4657644 0.89 ECE1 (0.52) ECE1CCR2
SCHEMBL4655305 0.89 ECE1 (0.46) ECE1CCR2MAPTTP53
SCHEMBL4655262 0.89 ECE1 (0.51) ECE1PPARGCCR9
SCHEMBL4656250 0.88 CACNA1H (0.49) ECE1CCR2MAPTTP53KDM4E
SCHEMBL15361984 0.87 MAOB (0.48) ECE1CCR2MAPTTP53KDM4E
Hydrochloric Acid SCHEMBL3576467 0.86 MAOB (0.47) ECE1CCR2MAPTTP53KDM4E
SCHEMBL3579347 0.86 ECE1 (0.51) ECE1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010297-B N- (1H-indolyl) -1H-indole-2-carboxamide derivatives, their preparation and their pharmaceutical use SANOFI AVENTIS 2011-07-27 CN claimed
EP-1776340-B1 N-(1H-INDOLYL)-H-INDOLE-2-CARB0XAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE SANOFI AVENTIS (FR) 2008-12-03 EP claimed