SCHEMBL4657644

SCHEMBL4657644

Cn1ccc2cc(NC(=O)c3cc4cc(F)ccc4n3Cc3ccccc3)ccc21

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 15/20 0.52
PTGDR2 Q9Y5Y4 2/20 0.49
NOTUM Q6P988 1/20 0.47
CCR2 P41597 1/20 0.47
ROCK1 Q13464 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579347 0.93 ECE1 (0.51) ECE1PTGDR2NOTUMCCR2
SCHEMBL4655305 0.92 ECE1 (0.46) ECE1PTGDR2NOTUMCCR2
SCHEMBL4655303 0.92 ECE1 (0.49) ECE1CCR2
SCHEMBL4656256 0.91 ECE1 (0.62) ECE1PTGDR2NOTUM
SCHEMBL4656230 0.91 ECE1 (0.60) ECE1PTGDR2NOTUMCCR2
SCHEMBL15361984 0.90 MAOB (0.48) ECE1PTGDR2CCR2
SCHEMBL4655328 0.90 PTGS2 (0.46) ECE1PTGDR2CCR2
Hydrochloric Acid SCHEMBL3576467 0.90 MAOB (0.47) ECE1PTGDR2CCR2
SCHEMBL4656147 0.90 ECE1 (0.55) ECE1PTGDR2NOTUM
SCHEMBL4655386 0.89 ECE1 (0.51) ECE1PTGDR2NOTUMCCR2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010297-B N- (1H-indolyl) -1H-indole-2-carboxamide derivatives, their preparation and their pharmaceutical use SANOFI AVENTIS 2011-07-27 CN claimed
EP-1776340-B1 N-(1H-INDOLYL)-H-INDOLE-2-CARB0XAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE SANOFI AVENTIS (FR) 2008-12-03 EP claimed