SCHEMBL4655419

SCHEMBL4655419

Cc1cc(C)cc(-n2c(C(=O)Nc3ccc4ccn(C)c4c3)cc3ccccc32)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.47
ECE1 P42892 1/20 0.43
GPX4 P36969 1/20 0.42
AHR P35869 1/20 0.42
GRM4 Q14833 1/20 0.42
MET P08581 1/20 0.41
THRB P10828 2/20 0.41
MAPT P10636 2/20 0.41
MAOB P27338 1/20 0.41
NOTUM Q6P988 1/20 0.41
ROR1 Q01973 1/20 0.40
TSHR P16473 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4655315 0.93 ECE1 (0.48) ECE1GPX4AHRGRM4MET
SCHEMBL4656242 0.84 ECE1 (0.49) ECE1GPX4METTHRBMAPT
SCHEMBL4656220 0.82 ECE1 (0.59) ECE1GPX4GRM4MAPTMAOB
SCHEMBL4655371 0.81 MDM2 (0.42) GRM4THRBMAPTTSHRALDH1A1
SCHEMBL4655332 0.80 MAPT (0.47) ECE1GPX4AHRGRM4MET
SCHEMBL4655241 0.80 NOTUM (0.49) ECE1GPX4METMAPTMAOB
SCHEMBL4655331 0.79 MAOB (0.51) ECE1GPX4GRM4METMAPT
SCHEMBL4655285 0.79 ECE1 (0.53) ECE1GPX4MAPTMAOBNOTUM
SCHEMBL4656319 0.79 ECE1 (0.50) ECE1GPX4AHRGRM4MET
SCHEMBL4655289 0.77 ECE1 (0.53) ECE1GPX4GRM4MAPTMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776340-B1 N-(1H-INDOLYL)-H-INDOLE-2-CARB0XAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE SANOFI AVENTIS (FR) 2008-12-03 EP claimed