SCHEMBL4656200

SCHEMBL4656200

O=[C]C1Cc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
KDM1A O60341 4/20 0.39
HTR2A P28223 3/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
SIGMAR1 Q99720 1/20 0.37
KMT2A Q03164 1/20 0.37
ANPEP P15144 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9160631 1.00 CHRNB2 (0.44) CHRNB2CHRNA4GRIN2DGRIN3BGRIN1
SCHEMBL9165647 0.78 IDO1 (0.46)
SCHEMBL384148 0.78 IDO1 (0.46)
SCHEMBL1722308 0.77 GRIN2D (0.41) CHRNB2CHRNA4GRIN2DGRIN3BGRIN1
SCHEMBL7431326 0.77 GRIN2D (0.41) CHRNB2CHRNA4GRIN2DGRIN3BGRIN1
SCHEMBL1756937 0.75 IDO1 (0.49) KMT2A
SCHEMBL9167813 0.75 IDO1 (0.49) KMT2A
SCHEMBL9159886 0.75 IDO1 (0.49) KMT2A
SCHEMBL2680028 0.72 S100A4 (0.41) HTR2CHTR2BKMT2A
SCHEMBL6649584 0.71 SLC6A2 (0.36) ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP claimed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US claimed
EP-1006122-A1 PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-06-07 EP claimed
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP disclosed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US disclosed
EP-1006122-A1 PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-06-07 EP disclosed