SCHEMBL4657144

SCHEMBL4657144

Cc1ccc([N+](=O)[O-])c(CCCC#N)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
CYP3A4 P08684 1/20 0.49
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
KAT2B Q92831 3/20 0.41
MAPT P10636 2/20 0.39
ACHE P22303 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658079 0.83 ALDH1A1 (0.41) TSHRCYP3A4ALDH1A1HPGDMAPT
SCHEMBL4656748 0.82 VCAM1 (0.49) TSHRALDH1A1HPGDMAPTNPC1
SCHEMBL16129051 0.81 ALDH1A1 (0.60) TSHRCYP3A4ALDH1A1HPGDKAT2B
SCHEMBL3636229 0.80 KAT2B (0.57) TSHRCYP3A4KAT2BACHENPC1
SCHEMBL2214742 0.80 ALDH1A1 (0.67) TSHRALDH1A1HPGDMAPTACHE
SCHEMBL27593715 0.77 MAPT (0.48) TSHRCYP3A4ALDH1A1HPGDMAPT
SCHEMBL4658987 0.77 NPC1 (0.49) TSHRCYP3A4ALDH1A1NPC1RAB9A
SCHEMBL4658092 0.77 TSHR (0.49) TSHRCYP3A4ALDH1A1KAT2BMAPT
SCHEMBL4966586 0.76 TSHR (0.56) TSHRCYP3A4ALDH1A1KAT2BMAPT
SCHEMBL27780345 0.76 TSHR (0.56) TSHRCYP3A4ALDH1A1KAT2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1295864-B1 PROCESS FOR PREPARATION OF 1,5-DIAMINONAPHTHALENES MITSUI CHEMICALS POLYURETHANES (JP) 2008-12-03 EP disclosed
US-6737548-B2 REACTING AN ORTHO-ALKYLNITROBENZENE WITH VINYL COMPOUND IN PRESENCE OF A BASE TO PRODUCE AN INTERMEDIATE, CYCLIZING THE INTERMEDIATE TO FORM 5-NITRO-1-TETRALONE COMPOUND, THEN REACTING WITH AMINE TO PRODUCE DIAMINONAPHTHALENE COMPOUNDS MITSUI CHEMICALS, INC. (JP) 2004-05-18 US disclosed
US-20030176722-A1 Process for preparation of 1,5-diaminonaphthalenes MITSUI CHEMICALS POLYURETHANES, INC. (JP) 2003-09-18 US disclosed
EP-1295864-A1 PROCESS FOR PREPARATION OF 1,5-DIAMINONAPHTHALENES Mitsui Chemicals, Inc. (JP) 2003-03-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030176722-A1 Process for preparation of 1,5-diaminonaphthalenes NOX5, NOX1, DPYD TSHR 4208/4885CYP3A4 154/4885ALDH1A1 159/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.