SCHEMBL4658121

SCHEMBL4658121

COC(Cc1ccccc1)(NC(C)=O)OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
RECQL P46063 2/20 0.55
MMP8 P22894 2/20 0.48
MAPT P10636 1/20 0.45
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
CTRB1 P17538 3/20 0.42
CYP1A2 P05177 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HIF1A Q16665 1/20 0.42
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPRA P18433 1/20 0.41
PTPRB P23467 1/20 0.41
MAPK1 P28482 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA3 P07451 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7959025 0.81 MEN1 (0.57) ALDH1A1SMN1; SMN2PTPN2PTPN1PTPRB
SCHEMBL6514301 0.77 ALDH1A1 (0.65) ALDH1A1RECQLMMP8MAPTCYP3A4
SCHEMBL28168069 0.75 ALDH1A1 (0.67) ALDH1A1RECQLMMP8MAPTCYP3A4
SCHEMBL25846939 0.75 ALDH1A1 (0.54) ALDH1A1RECQLMMP8MAPTCYP3A4
SCHEMBL27457092 0.74 ALDH1A1 (0.47) ALDH1A1RECQLMMP8CYP3A4CYP2C9
SCHEMBL6497301 0.74 TSHR (0.43) ALDH1A1RECQLMMP8CYP3A4CYP2C9
SCHEMBL8410894 0.74 ALDH1A1 (0.53) ALDH1A1RECQLMMP8MAPTCYP3A4
SCHEMBL8583261 0.74 ALDH1A1 (0.53) ALDH1A1RECQLMMP8CYP3A4CYP2C9
SCHEMBL2331138 0.74 ALDH1A1 (0.53) ALDH1A1RECQLMMP8MAPTCYP3A4
SCHEMBL2329888 0.74 ALDH1A1 (0.53) ALDH1A1RECQLMMP8MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996574-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES AS PHOSPHODIESTERASE 10 INHIBITORS Amgen Inc. (US) 2008-12-03 EP disclosed
WO-2007103554-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC. (US) 2007-09-13 WO disclosed