SCHEMBL7959025

SCHEMBL7959025

COC(Cc1ccccc1)(NC(=O)OCc1ccccc1)OC

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 1/20 0.48
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
PTPRB P23467 1/20 0.47
ACP1 P24666 1/20 0.47
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
CTSS P25774 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658121 0.81 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2LMNAPTPN2PTPN1
SCHEMBL6380611 0.80 MEN1 (0.57) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL4442846 0.79 KMT2A (0.60) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL10655573 0.79 ITGB3 (0.60) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL10654800 0.79 ITGB3 (0.60) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28199355 0.79 ITGB3 (0.60) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL843747 0.79 MEN1 (0.57) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL7271033 0.78 KMT2A (0.52) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28199962 0.78 MEN1 (0.52) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28199963 0.78 MEN1 (0.52) MEN1KMT2ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271238-B1 USEFUL IN TREATING AND PREVENTING DISEASES INVOLVING CHYMOTRYPSIN TYPE PROTEASES WHICH ARE RELATED TO ASTHMA, ALLERGY, INFLAMMATIONS, RHEUMATISM, HYPERTENSION, HEART FAILURE, MYOCARDIAL INFARCTION, AND CARDIAC HYPERTROPHY NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed
EP-0936216-A1 NOVEL ACETAMIDE DERIVATIVES AND PROTEASE INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1999-08-18 EP disclosed