Psi-6130-Tp

Psi-6130-Tp

SCHEMBL465832

C[C@@]1(F)[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(N)nc1=O

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 3/20 0.59
POLG P54098 2/20 0.57
P2RY2 P41231 10/20 0.55
P2RY4 P51582 6/20 0.55
PDE4D Q08499 1/20 0.51
PDE3A Q14432 1/20 0.51
SLC29A1 Q99808 1/20 0.51
POLB P06746 1/20 0.51
P2RY6 Q15077 5/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Psi-6130-Tp SCHEMBL12878130 1.00 POLA1 (0.59) POLA1POLGP2RY2P2RY4PDE4D
Psi-6130-Tp SCHEMBL12849776 1.00 POLA1 (0.59) POLA1POLGP2RY2P2RY4PDE4D
Psi-6130-Tp SCHEMBL21233069 1.00 POLA1 (0.59) POLA1POLGP2RY2P2RY4PDE4D
Psi-6130-Tp SCHEMBL12799368 1.00 POLA1 (0.59) POLA1POLGP2RY2P2RY4PDE4D
Psi-6130-Tp SCHEMBL15038016 1.00 POLA1 (0.59) POLA1POLGP2RY2P2RY4PDE4D
SCHEMBL12849778 0.98 POLA1 (0.61) POLA1POLGP2RY2P2RY4PDE4D
SCHEMBL12878128 0.98 POLA1 (0.61) POLA1POLGP2RY2P2RY4PDE4D
SCHEMBL12799372 0.98 POLA1 (0.61) POLA1POLGP2RY2P2RY4PDE4D
SCHEMBL471161 0.93 POLG (0.57) POLA1POLGP2RY2P2RY4PDE4D
Gemcitabine Triphosphate SCHEMBL3468704 0.91 POLA1 (0.69) POLA1POLGP2RY2P2RY4PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4032897-B1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES GILEAD PHARMASSET LLC (US) 2025-01-29 EP disclosed
EP-2604620-B9 Modified fluorinated nucleoside analogues GILEAD PHARMASSET LLC (US) 2024-10-23 EP disclosed
EP-2604620-B2 Modified fluorinated nucleoside analogues GILEAD PHARMASSET LLC (US) 2024-06-19 EP disclosed
EP-4032897-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES Gilead Pharmasset LLC (US) 2022-07-27 EP disclosed
EP-3521297-B1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES GILEAD PHARMASSET LLC (US) 2021-12-22 EP disclosed
US-20190315792-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, LTD. (BB) 2019-10-17 US disclosed
EP-3521297-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES Gilead Pharmasset LLC (US) 2019-08-07 EP disclosed
US-10287311-B2 Modified fluorinated nucleoside analogues GILEAD PHARMASSET LLC (US) 2019-05-14 US disclosed
EP-2604620-B1 Modified fluorinated nucleoside analogues GILEAD PHARMASSET LLC (US) 2016-06-29 EP disclosed
EP-2604620-A1 Modified fluorinated nucleoside analogues Gilead Pharmasset LLC (US) 2013-06-19 EP disclosed
EP-2345658-A1 Modified fluorinated nucleoside analogues Pharmasset, Inc. (US) 2011-07-20 EP disclosed
US-20110038833-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2011-02-17 US disclosed
US-20090036666-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2009-02-05 US disclosed
US-20090004135-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2009-01-01 US disclosed
US-20080253995-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2008-10-16 US disclosed
US-7429572-B2 Modified fluorinated nucleoside analogues PHARMASSET, INC. (US) 2008-09-30 US disclosed
US-20080070861-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2008-03-20 US disclosed
EP-1633766-A2 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES Pharmasset, Inc. (US) 2006-03-15 EP disclosed
WO-2005003147-A2 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES PHARMASSET, INC. (US) 2005-01-13 WO disclosed
US-20050009737-A1 Modified fluorinated nucleoside analogues GILEAD SCIENCES, INC. 2005-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080070861-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-10287311-B2 Modified fluorinated nucleoside analogues NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20090036666-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20190315792-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20050009737-A1 Modified fluorinated nucleoside analogues NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20110038833-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20090004135-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885
US-20080253995-A1 MODIFIED FLUORINATED NUCLEOSIDE ANALOGUES NSUN2, NT5C3B, METTL3 POLA1 2700/4885POLG 2915/4885P2RY2 378/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.