SCHEMBL4658573

SCHEMBL4658573

Cn1cc(C(=O)OCl)c2ccccc21

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.73
LMNA P02545 2/20 0.62
ALDH1A1 P00352 2/20 0.62
KMT2A Q03164 2/20 0.62
MITF O75030 1/20 0.62
MAPT P10636 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
POLB P06746 1/20 0.59
HTT P42858 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.52
RAB9A P51151 2/20 0.50
BRD4 O60885 1/20 0.50
UTS2R Q9UKP6 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.49
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28159208 0.89 NR4A2 (0.59) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL1092934 0.85 NR4A2 (1.00) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL31621504 0.85 NR4A2 (1.00) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL20554177 0.83 NR4A2 (0.73) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL28279140 0.83 NR4A2 (0.68) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL30958431 0.81 LMNA (0.68) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL2434450 0.81 LMNA (0.68) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL6379635 0.81 NR4A2 (0.69) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL17995258 0.81 NR4A2 (0.69) NR4A2LMNAALDH1A1KMT2AMITF
SCHEMBL5137040 0.80 NR4A2 (0.47) NR4A2LMNAALDH1A1KMT2AMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153643-A Substituted indole MCL-1 inhibitors 范德比尔特大学 2019-01-04 CN disclosed
EP-1917255-A2 INDOL-3-YL-CARBONYL-PIPERIDIN AND PIPERAZIN DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-05-07 EP disclosed
WO-2007014851-A2 INDOL-3-YL-CARBONYL-PIPERIDIN AND PIPERAZIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-02-08 WO disclosed