SCHEMBL4658705

SCHEMBL4658705

CC(C)(C)OC(=O)NN=C1CCOCC1.O=C1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 5/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.38
CTSK P43235 2/20 0.36
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.35
MIF P14174 1/20 0.35
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
USP2 O75604 1/20 0.34
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1406859 0.94 KMT2A (0.58) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL17525371 0.85 KMT2A (0.52) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL14990248 0.85 KMT2A (0.52) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL11947773 0.85 KMT2A (0.52) KMT2AALDH1A1KDM4EMAPTMEN1
Hydrochloric Acid SCHEMBL4657741 0.80 KMT2A (0.52) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL573354 0.79 ALDH1A1 (0.63) KMT2AALDH1A1KDM4ERAB9AMIF
SCHEMBL272269 0.79 ALDH1A1 (0.63) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL3490122 0.78 ALDH1A1 (0.58) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL182243 0.78 ALDH1A1 (0.61) KMT2AALDH1A1KDM4EMEN1LMNA
SCHEMBL20583517 0.78 KMT2A (0.54) KMT2AALDH1A1KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999114-A2 PYRAZOLES AS 11-BETA-HSD-1 F. Hoffmann-la Roche AG (CH) 2008-12-10 EP disclosed
WO-2007107470-A2 PYRAZOLES AS 11-BETA-HSD-1 F. HOFFMANN-LA ROCHE AG (CH) 2007-09-27 WO disclosed