SCHEMBL4658992

SCHEMBL4658992

CNC1=NCC(c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MAPT P10636 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
RECQL P46063 1/20 0.40
HSD17B10 Q99714 1/20 0.40
OPRK1 P41145 1/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
BCHE P06276 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701530 0.83 TERT (0.39) HTR2AHTR2CHTR2BHRH3MAPT
Hydrochloric Acid SCHEMBL702047 0.82 TERT (0.39) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL28808620 0.70 HTR2A (0.44) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL28628435 0.68 HTR2A (0.57) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL702690 0.66 HTR2A (0.38) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL701484 0.65 MEN1 (0.38) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL702297 0.65 MAPT (0.36) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL9149487 0.64 HTR2A (0.49) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL11018166 0.63 HTR2A (0.48) HTR2AHTR2CHTR2BHRH3MAPT
SCHEMBL22335132 0.63 NPC1 (0.57) MAPTSMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999113-A1 SUBSTITUTED 1-AMINO-4-PHENYL-DIHYDROISOQUINOLINES, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF AS A MEDICAMENT, AND MEDICAMENTS CONTAINING THEM Sanofi-Aventis (FR) 2008-12-10 EP disclosed
WO-2007107245-A1 SUBSTITUTED 1-AMINO-4-PHENYL-DIHYDROISOQUINOLINES, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF AS A MEDICAMENT, AND MEDICAMENTS CONTAINING THEM SANOFI-AVENTIS (FR) 2007-09-27 WO disclosed