SCHEMBL4659280

SCHEMBL4659280

CC(C)c1cc2c(cc1N1C[C@@H](CN)OC1=O)NC(=O)C2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.36
SMYD3 Q9H7B4 8/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
GRM2 Q14416 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5499874 0.86 F10 (0.39) F10GRIA1CACNG8GRM2
SCHEMBL5499028 0.84 F10 (0.37) F10SMYD3GRIA1CACNG8GRM2
SCHEMBL5501644 0.79 F10 (0.35) F10GRIA1CACNG8GRM2
SCHEMBL5502999 0.79 F10 (0.37) F10SMYD3GRIA1CACNG8
SCHEMBL5502470 0.79 F10 (0.37) F10SMYD3GRIA1CACNG8
SCHEMBL5499114 0.78 SMYD3 (0.34) SMYD3LMNAGAAGRIA1CACNG8
SCHEMBL5502896 0.78 F10 (0.36) F10SMYD3GRIA1CACNG8GRM2
SCHEMBL5502616 0.77 F10 (0.35) F10SMYD3
SCHEMBL5506392 0.76 GRM2 (0.36) F10GRM2
SCHEMBL5499076 0.71 GRM2 (0.37) F10GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004640-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS Pfizer Products Inc. (US) 2008-12-24 EP disclosed
EP-1869029-A1 AN OXINDOLE OXAZOLIDINONE AS ANTIBACTERIAL AGENT Pharmacia & Upjohn Company LLC (US) 2007-12-26 EP disclosed
WO-2007091147-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS PFIZER PRODUCTS INC. (US) 2007-08-16 WO disclosed
WO-2006106426-A1 AN OXINDOLE OXAZOLIDINONE AS ANTIBACTERIAL AGENT PHARMACIA & UPJOHN COMPANY LLC (US) 2006-10-12 WO disclosed