SCHEMBL4659730

SCHEMBL4659730

CC(C)(C)c1ccc(S(=O)(=O)N(Cc2ccccc2)c2ccc3[nH]c(OC(=O)NC4CCOCC4)c(-c4ccccc4)c3c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.37
PTGES O14684 3/20 0.36
ALOX5 P09917 2/20 0.36
RORC P51449 3/20 0.36
PTPN22 Q9Y2R2 5/20 0.36
NR3C1 P04150 2/20 0.36
PTPN1 P18031 2/20 0.35
PTPN12 Q05209 2/20 0.35
TRPM8 Q7Z2W7 1/20 0.34
OXTR P30559 1/20 0.34
AVPR1A P37288 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4762894 0.89 TP53 (0.36) HTT
SCHEMBL5151373 0.88 CA1 (0.41) MCL1PTGESALOX5RORCPTPN22
SCHEMBL4762138 0.85 MCL1 (0.45) MCL1PTGESALOX5RORCPTPN22
SCHEMBL4792514 0.83 MCL1 (0.41) MCL1PTGESALOX5RORCPTPN22
SCHEMBL4762404 0.82 BRD4 (0.42)
SCHEMBL3947584 0.82 BRD4 (0.48)
SCHEMBL5151586 0.80 CA1 (0.40) MCL1RORCOXTRAVPR1AGAA
SCHEMBL4762136 0.78 MCL1 (0.49) MCL1PTGESALOX5RORCPTPN22
SCHEMBL5149450 0.77 CA1 (0.42) GAAHTT
SCHEMBL3941796 0.76 BRD4 (0.43) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001847-A2 SOLUBLE ADENYLATE CYCLASE INHIBITORS Bayer Schering Pharma AG (DE) 2008-12-17 EP claimed
WO-2007107385-A2 SOLUBLE ADENYLATE CYCLASE INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-09-27 WO claimed
EP-2001847-A2 SOLUBLE ADENYLATE CYCLASE INHIBITORS Bayer Schering Pharma AG (DE) 2008-12-17 EP disclosed
WO-2007107385-A2 SOLUBLE ADENYLATE CYCLASE INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-09-27 WO disclosed