SCHEMBL4659840

SCHEMBL4659840

CS(=O)(=O)Nc1ccc(-c2ccc(C(F)(F)F)cc2)cc1F

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 14/20 0.74
SLC22A12 Q96S37 1/20 0.53
TRPV1 Q8NER1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661054 0.86 KIF11 (0.56) KIF11SLC22A12TRPV1
SCHEMBL4659833 0.85 KIF11 (0.74) KIF11
SCHEMBL5529232 0.85 KIF11 (1.00) KIF11
SCHEMBL4661102 0.85 KIF11 (0.76) KIF11SLC22A12
SCHEMBL4659924 0.84 KIF11 (0.74) KIF11SLC22A12TRPV1
SCHEMBL4661499 0.84 KIF11 (0.76) KIF11SLC22A12
SCHEMBL4661117 0.83 KIF11 (0.73) KIF11SLC22A12
SCHEMBL4661120 0.83 TRPV1 (0.54) KIF11SLC22A12TRPV1
SCHEMBL3376561 0.80 KIF11 (0.61) KIF11SLC22A12
SCHEMBL4661073 0.80 KIF11 (0.76) KIF11SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694281-A4 BIPHENYL COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2008-12-24 EP claimed
US-20070259951-A1 Compounds, Compositions and Methods SMITHKLINE BEECHAM CORPORATION (US) 2007-11-08 US claimed
EP-1694281-A2 BIPHENYL COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-08-30 EP claimed
WO-2005060692-A2 BIPHENYL COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-07 WO claimed
US-20070259951-A1 Compounds, Compositions and Methods SMITHKLINE BEECHAM CORPORATION (US) 2007-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070259951-A1 Compounds, Compositions and Methods ALPP, PCNA, MKI67 KIF11 824/4885SLC22A12 3290/4885TRPV1 4639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.