SCHEMBL4664520

SCHEMBL4664520

C=C(C)C(=O)OCC(C)(C)c1cc(-n2nc3ccc(Cl)cc3n2)c(O)c(C(C)(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664025 0.89 NPC1 (0.36) NPC1RAB9A
SCHEMBL4666346 0.88 XPO1 (0.32)
SCHEMBL1973788 0.85 RXFP1 (0.33) NPC1RAB9A
SCHEMBL4664022 0.84 CNR2 (0.32)
SCHEMBL29384523 0.83 GAA (0.31) NPC1RAB9A
SCHEMBL93350 0.83 GAA (0.31) NPC1RAB9A
SCHEMBL4664015 0.83
SCHEMBL4667550 0.83 NPC1 (0.32) NPC1RAB9A
SCHEMBL227535 0.82 GAA (0.33)
SCHEMBL29370220 0.82 GAA (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1949144-A2 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2008-07-30 EP claimed
WO-2007050395-A2 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2007-05-03 WO claimed
US-20070092831-A1 Radiation-absorbing polymeric materials and ophthalmic devices comprising same BAUSCH & LOMB INCORPORATED 2007-04-26 US claimed
WO-2006119304-A1 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2006-11-09 WO claimed
US-20060252850-A1 Radiation-absorbing polymeric materials and ophthalmic devices comprising same BAUSCH & LOMB INCORPORATED 2006-11-09 US claimed
EP-3174940-B1 ULTRAVIOLET-CURABLE COATING AGENT WITH IMPROVED SUNLIGHT RESISTANCE TIGER COATINGS GMBH & CO KG (AT) 2019-02-06 EP disclosed
US-20170260399-A1 UV-Curable Coating Composition Having Improved Sunlight Stability TIGER COATINGS GMBH & CO. KG (AT) 2017-09-14 US disclosed
EP-3174940-A1 UV-CURABLE COATING COMPOSITION HAVING IMPROVED SUNLIGHT STABILITY TIGER Coatings GmbH & Co. KG (AT) 2017-06-07 EP disclosed
WO-2016016112-A1 UV-CURABLE COATING COMPOSITION HAVING IMPROVED SUNLIGHT STABILITY TIGER COATINGS GMBH & CO. KG (AT) 2016-02-04 WO disclosed
EP-1949144-A2 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2008-07-30 EP disclosed
WO-2007050395-A2 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2007-05-03 WO disclosed
WO-2007050394-A2 POLYMERIC RADIATION-ABSORBING MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2007-05-03 WO disclosed
US-20070092831-A1 Radiation-absorbing polymeric materials and ophthalmic devices comprising same BAUSCH & LOMB INCORPORATED 2007-04-26 US disclosed
US-20070092830-A1 Polymeric radiation-absorbing materials and ophthalmic devices comprising same BAUSCH & LOMB INCORPORATED 2007-04-26 US disclosed
WO-2006119304-A1 RADIATION-ABSORBING POLYMERIC MATERIALS AND OPHTHALMIC DEVICES COMPRISING SAME BAUSCH & LOMB INCORPORATED (US) 2006-11-09 WO disclosed
US-20060252850-A1 Radiation-absorbing polymeric materials and ophthalmic devices comprising same BAUSCH & LOMB INCORPORATED 2006-11-09 US disclosed