SCHEMBL4665871

SCHEMBL4665871

COC(=O)c1cc(OC)ccc1Nc1cc(C(C)(C)C)nn1-c1cnccc1C

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.46
BRAF P15056 1/20 0.46
MAPK14 Q16539 14/20 0.44
PTK2 Q05397 1/20 0.42
PTK2B Q14289 1/20 0.42
MAPK12 P53778 6/20 0.41
MAPK13 O15264 4/20 0.41
MAPK11 Q15759 3/20 0.41
ADORA1 P30542 3/20 0.41
HCK P08631 2/20 0.40
SRC P12931 2/20 0.40
GSK3A P49840 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600184 0.93 ADORA1 (0.49) RAF1BRAFMAPK14PTK2PTK2B
SCHEMBL5008532 0.89 MAPK14 (0.47) MAPK14PTK2PTK2BMAPK12MAPK13
SCHEMBL5008723 0.83 MAPK14 (0.46) MAPK14PTK2PTK2BMAPK12MAPK13
SCHEMBL4667080 0.81 GFER (0.57) ADORA1
SCHEMBL5012222 0.80 ADORA1 (0.62) MAPK14MAPK12MAPK13MAPK11ADORA1
SCHEMBL14600217 0.80 MAPK14 (0.50) RAF1BRAFMAPK14MAPK12MAPK13
SCHEMBL5008440 0.79 MAPK14 (0.45) MAPK14PTK2PTK2BMAPK12MAPK13
SCHEMBL5008388 0.79 MAPK14 (0.53) BRAFMAPK14MAPK12MAPK13MAPK11
SCHEMBL5007711 0.79 MAPK14 (0.47) RAF1MAPK14MAPK12MAPK13MAPK11
SCHEMBL14600243 0.78 GFER (0.53) MAPK14PTK2MAPK12MAPK13MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed