SCHEMBL4666774

SCHEMBL4666774

N#Cc1ccccc1Cc1c[nH]nn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.37
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
ALDH1A1 P00352 5/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PLAU P00749 1/20 0.35
ALOX15 P16050 1/20 0.35
ATM Q13315 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CNR2 P34972 1/20 0.34
KDM4E B2RXH2 2/20 0.34
TP53 P04637 1/20 0.34
BCAT2 O15382 1/20 0.34
HPGD P15428 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12468870 0.75 IDO1 (0.40) CYP19A1ALDH1A1NPC1RAB9AKDM4E
SCHEMBL28758851 0.75 IDO1 (0.44) ALDH1A1
SCHEMBL27164548 0.74 ALDH1A1 (0.39) CYP19A1SMN1; SMN2TLR8TLR7ALDH1A1
SCHEMBL2153612 0.74 CYP19A1 (0.48) CYP19A1SMN1; SMN2ALDH1A1MAPTNPC1
SCHEMBL2825597 0.72 DPP4 (0.43) SLC6A4
SCHEMBL2727911 0.71 CYP19A1 (0.45) CYP19A1SMN1; SMN2ALDH1A1MAPTALOX15
SCHEMBL11294215 0.71 ALDH1A1 (0.40) CYP19A1ALDH1A1MAPTSLC6A4
SCHEMBL1931499 0.70 HSPA5 (0.37) SMN1; SMN2ALDH1A1MAPTALOX15HSD17B10
SCHEMBL27164067 0.70 TSHR (0.39) CYP19A1SMN1; SMN2ALDH1A1MAPTPLAU
SCHEMBL2903299 0.69 HRH3 (0.50) CYP19A1TLR8TLR7ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871750-A1 IMPROVED PROCESS FOR THE PREPARATION OF LETROZOLE Sicor, Inc. (US) 2008-01-02 EP claimed
WO-2007100346-A1 IMPROVED PROCESS FOR THE PREPARATION OF LETROZOLE SICOR, INC. (US) 2007-09-07 WO claimed