SCHEMBL2903299

SCHEMBL2903299

N#Cc1cccc(Cc2c[nH]nn2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.50
MPO P05164 1/20 0.45
GLA P06280 1/20 0.42
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
ALDH1A1 P00352 3/20 0.40
SLC6A4 P31645 2/20 0.39
DAO P14920 1/20 0.39
IDH1 O75874 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
SLC6A2 P23975 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767382 0.81 HRH3 (0.45) HRH3CYP19A1DAOKMT2A
SCHEMBL31132412 0.76 HTR1B (0.45) IDH1GABRG2GABRB3GABRA3MAPT
SCHEMBL28758849 0.76 IDO1 (0.43) CYP11B1CYP11B2
SCHEMBL2153847 0.76 HRH3 (0.59) HRH3MPOGLACYP19A1CYP11B1
SCHEMBL29272 0.75 ALDH1A1 (0.46) HRH3ALDH1A1MAPTMEN1TSHR
Benzene SCHEMBL27499662 0.75 ALDH1A1 (0.46) HRH3ALDH1A1MAPTMEN1TSHR
SCHEMBL28758850 0.74 HTR1B (0.50) DAO
SCHEMBL22968664 0.74 HRH3 (0.55) HRH3MPOGLACYP19A1CYP11B1
SCHEMBL29467167 0.74 HRH3 (0.55) HRH3MPOGLACYP19A1CYP11B1
SCHEMBL9508013 0.73 ALDH1A1 (0.44) HRH3ALDH1A1MAPTMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212301-A1 AN IMPROVED PROCESS FOR PREPARATION OF LETROZOLE AND ITS INTERMEDIATES Fresenius Kabi Oncology Limited (IN) 2010-08-04 EP disclosed
WO-2009069140-A1 AN IMPROVED PROCESS FOR PREPARATION OF LETROZOLE AND ITS INTERMEDIATES DABUR PHARMA LIMITED (IN) 2009-06-04 WO disclosed