SCHEMBL4667046

SCHEMBL4667046

CCc1nn(-c2cnccc2C)c(Nc2ccc(Cl)cc2C(=O)O)c1-c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 17/20 0.52
ADORA3 P0DMS8 1/20 0.40
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
ADORA2B P29275 1/20 0.38
KDM4C Q9H3R0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668528 0.92 ADORA1 (0.53) ADORA1ADORA3
SCHEMBL4668225 0.89 ADORA1 (0.44) ADORA1FABP3FABP4ADORA2BKDM4C
SCHEMBL4668016 0.84 ADORA1 (0.53) ADORA1ADORA3KDM4C
SCHEMBL4667055 0.80 ADORA1 (0.53) ADORA1ADORA3ADORA2B
SCHEMBL4666257 0.80 ADORA1 (0.48) ADORA1ADORA3
SCHEMBL4666092 0.80 ADORA1 (0.46) ADORA1FABP3FABP4ADORA2BKDM4C
SCHEMBL14600200 0.79 ADORA1 (0.51) ADORA1ADORA3ADORA2B
SCHEMBL4666215 0.79 ADORA1 (0.51) ADORA1ADORA3
Trifluoroacetic Acid SCHEMBL5007734 0.79 ADORA1 (0.67) ADORA1ADORA3ADORA2B
SCHEMBL14600708 0.78 ADORA1 (0.50) ADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed