SCHEMBL4667145

SCHEMBL4667145

O=C(O)CC(Cc1csc2ccccc12)NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.49
CASP1 P29466 1/20 0.48
KMT2A Q03164 2/20 0.43
MDM4 O15151 1/20 0.41
TP53 P04637 1/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
SLC17A5 Q9NRA2 1/20 0.41
POLB P06746 1/20 0.40
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667142 1.00 CASP3 (0.49) CASP3CASP1KMT2AMDM4TP53
SCHEMBL799761 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL29444635 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL29511478 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL6790172 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL3725892 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL30182933 0.86 MDM4 (0.51) CASP3CASP1MDM4TP53CTSL
SCHEMBL118132 0.84 CASP3 (0.53) CASP3CASP1KMT2AMDM4TP53
SCHEMBL4667137 0.84 CASP3 (0.53) CASP3CASP1KMT2AMDM4TP53
SCHEMBL118115 0.84 CASP3 (0.53) CASP3CASP1KMT2AMDM4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1985612-A1 Arymethylen substituted N-Acyl-gamma-aminoalcohols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-10-29 EP disclosed