SCHEMBL29444635

SCHEMBL29444635

O=C(N[C@@H](Cc1csc2ccccc12)C(=O)O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 3/20 0.51
TP53 P04637 3/20 0.51
CTSL P07711 1/20 0.48
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
SLC17A5 Q9NRA2 1/20 0.47
CASP1 P29466 1/20 0.47
CASP3 P42574 2/20 0.46
MDM2 Q00987 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30182933 1.00 MDM4 (0.51) MDM4TP53CTSLCTSSCTSK
SCHEMBL29511478 1.00 MDM4 (0.51) MDM4TP53CTSLCTSSCTSK
SCHEMBL6790172 1.00 MDM4 (0.51) MDM4TP53CTSLCTSSCTSK
SCHEMBL799761 1.00 MDM4 (0.51) MDM4TP53CTSLCTSSCTSK
SCHEMBL3725892 1.00 MDM4 (0.51) MDM4TP53CTSLCTSSCTSK
SCHEMBL6019567 0.87 CTSS (0.68) CTSLCTSSCTSK
SCHEMBL4667145 0.86 CASP3 (0.49) MDM4TP53CTSLCTSSCTSK
SCHEMBL4667142 0.86 CASP3 (0.49) MDM4TP53CTSLCTSSCTSK
SCHEMBL6019561 0.84 CTSL (0.49) MDM4TP53CTSLCTSSCTSK
SCHEMBL6019553 0.84 CTSL (0.53) MDM4TP53CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115068469-B TIGIT inhibitors and uses thereof 深圳市小分子新药创新中心有限公司 2024-02-27 CN disclosed
CN-115068469-A TIGIT inhibitor and application thereof 深圳市小分子新药创新中心有限公司 2022-09-20 CN disclosed
CN-113912670-B Angiotensin converting enzyme 2 inhibitor, application thereof and anti-coronavirus infection drug 深圳市小分子新药创新中心有限公司 2022-04-08 CN disclosed