SCHEMBL4668519

SCHEMBL4668519

CC(C)(C)Cc1cc(CC(CO)CCc2ccc(C(=O)O)cc2)ccc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
ACE2 Q9BYF1 2/20 0.37
GRIN2D O15399 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
BRS3 P32247 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
RARB P10826 4/20 0.34
FOLH1 Q04609 2/20 0.34
ADRB3 P13945 2/20 0.33
ADRB1 P08588 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PTGER4 P35408 1/20 0.33
PTGER2 P43116 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17965451 0.83 TSHR (0.39) TSHRGRIN2DGRIN2AGRIN2BGRIN2C
SCHEMBL3484562 0.83 RARB (0.43) TSHRACE2GRIN2DGRIN2AGRIN2B
SCHEMBL2489653 0.78 ANPEP (0.47) TSHRRARBFOLH1ALDH1A1PTGER4
SCHEMBL3484567 0.78 NR1H4 (0.41) TSHRACE2GRIN2DGRIN2AGRIN2B
SCHEMBL1618045 0.75 TDP1 (0.46) TSHRACE2TDP1NR1H4
SCHEMBL2160396 0.74 ALDH1A1 (0.48) TSHRTDP1RARBFOLH1ALDH1A1
Ethylene SCHEMBL9718947 0.73 TDP1 (0.44) TSHRACE2TDP1NR1H4
SCHEMBL3485094 0.71 NR1H4 (0.41) GRIN2DGRIN2AGRIN2BGRIN2CRARB
SCHEMBL3485088 0.70 SLC7A5 (0.40) ADRB3ADRB1NR1H4
Benzoic Acid SCHEMBL19874935 0.67 ADRB3 (0.49) TSHRFOLH1ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940769-B1 DICARBOXYLIC ACID DERIVATIVES AND THEIR USE BAYER IP GMBH (DE) 2016-08-10 EP disclosed
EP-1940769-A1 DICARBOXYLIC ACID DERIVATIVES AND THEIR USE Bayer HealthCare AG (DE) 2008-07-09 EP disclosed
WO-2007045433-A1 DICARBOXYLIC ACID DERIVATIVES AND THEIR USE BAYER HEALTHCARE AG (DE) 2007-04-26 WO disclosed