SCHEMBL4669408

SCHEMBL4669408

CNC(=O)OC1(CN(C=O)c2cccnc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
NOTUM Q6P988 1/20 0.34
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
HDAC6 Q9UBN7 2/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2B6 P20813 1/20 0.32
CYP2C19 P33261 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4825426 0.73 HTT (0.40) HTTNOTUMMAPTGFERNPSR1
SCHEMBL4669407 0.71 PTGIR (0.35) HTTNOTUMNPSR1TRPV1L3MBTL1
SCHEMBL4824840 0.70 GAA (0.44) HTTMAPTHDAC6GAAALDH1A1
SCHEMBL1850567 0.70 HTT (0.46) HTTNOTUMMAPTGFERNPSR1
SCHEMBL10502805 0.66 KCNA5 (0.41) HTTNOTUMMAPTGFERNPSR1
SCHEMBL25752263 0.64 HTT (0.55) HTTNOTUMMAPTGFERNPSR1
SCHEMBL10502630 0.63 KCNA5 (0.40) HTTNOTUMTRPV1L3MBTL1CYP3A4
SCHEMBL10650461 0.62 TBXAS1 (0.52)
SCHEMBL26957589 0.62 NOTUM (0.51) HTTNOTUMTRPV1GAAHPGD
Hydrochloric Acid SCHEMBL11775309 0.61 GAA (0.50) HTTMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1757586-B1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG SERVIER LAB (FR) 2008-12-03 EP disclosed
EP-1757586-A1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG Les Laboratoires Servier (FR) 2007-02-28 EP disclosed