SCHEMBL4669532

SCHEMBL4669532

COc1ccc2c(c1)CCNC2c1cc(Cl)cc(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.62
CA2 P00918 5/20 0.62
CA9 Q16790 5/20 0.62
CA14 Q9ULX7 5/20 0.62
CA7 P43166 4/20 0.62
GID4 Q8IVV7 1/20 0.55
KDM1A O60341 3/20 0.54
HTR2C P28335 3/20 0.51
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
PRCP P42785 1/20 0.44
CYP19A1 P11511 1/20 0.44
HTR2A P28223 2/20 0.43
HTR2B P41595 2/20 0.43
HTR1A P08908 1/20 0.43
DRD4 P21917 1/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28742350 0.89 CA1 (0.69) CA1CA2CA9CA14CA7
SCHEMBL5522656 0.83 GID4 (0.69) CA1CA2CA9CA14CA7
SCHEMBL5523066 0.82 CA1 (0.57) CA1CA2CA9CA14CA7
SCHEMBL4674453 0.82 KMT2A (0.71) CA1CA2CA9CA14CA7
SCHEMBL4242796 0.82 CA1 (0.60) CA1CA2CA9CA14CA7
SCHEMBL29670244 0.82 CA1 (0.70) CA1CA2CA9CA14CA7
SCHEMBL19453945 0.82 CA1 (0.70) CA1CA2CA9CA14CA7
SCHEMBL4244900 0.82 CA1 (0.54) CA1CA2CA9CA14CA7
SCHEMBL6716383 0.81 CA1 (0.69) CA1CA2CA9CA14CA7
SCHEMBL6715368 0.81 CA1 (0.69) CA1CA2CA9CA14CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732898-B1 TETRAHYDROISOQUINOLINE- AND TETRAHYDROBENZAZEPINE DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2008-01-23 EP disclosed