SCHEMBL4669747

SCHEMBL4669747

COc1ccc2c(c1)CCN(C)C2c1cc(Cl)cc(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.56
CA2 P00918 9/20 0.56
CA9 Q16790 9/20 0.56
CA14 Q9ULX7 9/20 0.56
DRD1 P21728 6/20 0.53
DRD2 P14416 5/20 0.48
DRD4 P21917 2/20 0.48
CA7 P43166 1/20 0.47
DRD5 P21918 2/20 0.44
DRD3 P35462 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4671145 0.92 CA1 (0.51) CA1CA2CA9CA14DRD1
SCHEMBL28742357 0.90 CA1 (0.69) CA1CA2CA9CA14DRD1
SCHEMBL4673775 0.83 DRD1 (0.52) CA1CA2CA9CA14DRD1
SCHEMBL28742343 0.83 CA1 (0.68) CA1CA2CA9CA14DRD1
SCHEMBL985863 0.83 CA1 (0.55) CA1CA2CA9CA14DRD1
SCHEMBL987287 0.83 CA1 (0.52) CA1CA2CA9CA14DRD1
Hydrochloric Acid SCHEMBL4674113 0.83 CA1 (0.52) CA1CA2CA9CA14DRD1
SCHEMBL985641 0.82 CA1 (0.54) CA1CA2CA9CA14DRD1
SCHEMBL8024197 0.76 MAOA (0.60) CA1CA2CA9CA14DRD1
Hydrochloric Acid SCHEMBL4674943 0.75 DRD1 (0.47) CA1CA2CA9CA14DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732898-B1 TETRAHYDROISOQUINOLINE- AND TETRAHYDROBENZAZEPINE DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2008-01-23 EP disclosed