SCHEMBL4673775

SCHEMBL4673775

COc1ccc2c(c1)CCN(C)C2c1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.52
CA1 P00915 8/20 0.48
CA2 P00918 8/20 0.48
CA9 Q16790 8/20 0.48
CA14 Q9ULX7 8/20 0.48
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
CA7 P43166 1/20 0.46
GRIN2D O15399 4/20 0.46
GRIN3B O60391 4/20 0.46
GRIN1 Q05586 4/20 0.46
GRIN2A Q12879 4/20 0.46
GRIN2B Q13224 4/20 0.46
GRIN2C Q14957 4/20 0.46
GRIN3A Q8TCU5 4/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4674943 0.91 DRD1 (0.47) DRD1CA1CA2CA9CA14
SCHEMBL4412560 0.84 MAOA (0.58) DRD1DRD2
SCHEMBL7911741 0.84 MAOA (0.58) DRD1DRD2
SCHEMBL4415052 0.84 MAOA (0.58) DRD1DRD2
SCHEMBL30799251 0.84 MAOA (0.58) DRD1DRD2
SCHEMBL4669747 0.83 CA1 (0.56) DRD1CA1CA2CA9CA14
SCHEMBL986382 0.83 CA1 (0.48) DRD1CA1CA2CA9CA14
SCHEMBL985708 0.83 DRD1 (0.48) DRD1CA1CA2CA9CA14
SCHEMBL985355 0.82 TSHR (0.58) DRD1CA1CA2CA9CA14
SCHEMBL28742343 0.82 CA1 (0.68) DRD1CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732898-B1 TETRAHYDROISOQUINOLINE- AND TETRAHYDROBENZAZEPINE DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2008-01-23 EP disclosed