SCHEMBL4670628

SCHEMBL4670628

NC(=O)c1ccc(N2CCN(CCCC3CCCC3)C2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.51
ADRB2 P07550 2/20 0.41
ADRB1 P08588 2/20 0.41
ADRB3 P13945 2/20 0.41
PARP15 Q460N3 3/20 0.41
PARP10 Q53GL7 3/20 0.41
DRD2 P14416 4/20 0.41
DRD3 P35462 4/20 0.41
S1PR1 P21453 1/20 0.40
OPRM1 P35372 3/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 1/20 0.39
PARP2 Q9UGN5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4670487 0.86 DRD2 (0.45) HDAC1ADRB2ADRB1ADRB3DRD2
SCHEMBL4670081 0.74 ADRB2 (0.42) ADRB2ADRB1ADRB3PARP15PARP10
SCHEMBL4670126 0.74 ADRB2 (0.41) ADRB2ADRB1ADRB3PARP15PARP10
Water SCHEMBL4673066 0.73 ADRB2 (0.41) ADRB2ADRB1ADRB3PARP15PARP10
SCHEMBL4670057 0.73 PARP15 (0.42) ADRB2ADRB1ADRB3PARP15PARP10
SCHEMBL4670413 0.73 PARP15 (0.42) ADRB2ADRB1ADRB3PARP15PARP10
Water SCHEMBL4672106 0.73 ADRB2 (0.41) ADRB2ADRB1ADRB3PARP15PARP10
SCHEMBL6301319 0.71 PARP10 (0.41) ADRB2ADRB1ADRB3PARP15PARP10
SCHEMBL4670624 0.71 PARP15 (0.40) ADRB2ADRB1ADRB3PARP15PARP10
Hydrochloric Acid SCHEMBL7392932 0.70 S1PR1 (0.51) HDAC1ADRB2ADRB1ADRB3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed
US-6051586-A HYPOGLYCEMIC AGENTS; ANTIDIABETIC AGENTS BAYER CORPORATION (US) 2000-04-18 US disclosed