SCHEMBL4670793

SCHEMBL4670793

Fc1cc2c(F)cccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.56
DDO Q99489 1/20 0.56
FLT3 P36888 2/20 0.44
HRH4 Q9H3N8 2/20 0.43
PDE7A Q13946 1/20 0.40
ALDH1A1 P00352 2/20 0.39
GPR3 P46089 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AHR P35869 1/20 0.38
KDM4E B2RXH2 2/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
ALB P02768 4/20 0.36
IL2 P60568 4/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
HPGD P15428 2/20 0.36
RAB9A P51151 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27739684 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL3632451 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL4692767 0.78 DAO (0.53) DAODDOFLT3HRH4ALDH1A1
SCHEMBL27889601 0.78 DAO (0.62) DAODDOFLT3HRH4PDE7A
SCHEMBL20005057 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL25142137 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL28813362 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL15951255 0.78 DAO (0.53) DAODDOFLT3HRH4PDE7A
SCHEMBL30605955 0.78 DAO (0.53) DAODDOFLT3HRH4ALDH1A1
SCHEMBL28251861 0.78 DAO (0.53) DAODDOFLT3HRH4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173432-B9 PIPERIDINE-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY NPS ALLELIX CORP (CA) 2008-10-15 EP disclosed
EP-1173432-B1 PIPERIDINE-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY NPS ALLELIX CORP (CA) 2007-10-17 EP disclosed
US-6133287-A SEROTONIN 5-HT6 RECEPTOR ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS, E.G., PSYCHOSIS, SCHIZOPHRENIA, MANIC DEPRESSION, DEPRESSION, MEMORY DISTURBANCES, PARKINSONISM, AMYLOTROPHIC LATERAL SCLEROSIS, ALZHEIMER'S AND HUNTINGTON'S DISEASE ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-10-17 US disclosed