SCHEMBL4671797

SCHEMBL4671797

O=C(Cc1cccc(Cl)c1)NCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1.O=C(Cc1ccccc1Nc1c(Cl)cccc1Cl)NCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.44
AVPR1A P37288 3/20 0.44
EPHX2 P34913 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA9 Q16790 1/20 0.42
MAPT P10636 2/20 0.41
MAPK1 P28482 1/20 0.41
CCR2 P41597 1/20 0.41
CXCR6 O00574 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
AKR1B10 O60218 1/20 0.40
UGT1A9 O60656 1/20 0.40
TRPA1 O75762 1/20 0.40
ABCB11 O95342 1/20 0.40
MT-CO2 P00403 1/20 0.40
TTR P02766 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4671794 1.00 SIGMAR1 (0.44) SIGMAR1AVPR1AEPHX2CA12CA1
SCHEMBL3870289 0.94 AVPR1A (0.46) SIGMAR1AVPR1ACA12CA1CA2
SCHEMBL3870291 0.94 AVPR1A (0.46) SIGMAR1AVPR1ACA12CA1CA2
SCHEMBL3871878 0.89 AVPR1A (0.50) SIGMAR1AVPR1ACA12CA1CA2
SCHEMBL3871881 0.89 AVPR1A (0.50) SIGMAR1AVPR1ACA12CA1CA2
SCHEMBL3869562 0.88 EPHX2 (0.54) SIGMAR1AVPR1AEPHX2MAPTMAPK1
SCHEMBL3869565 0.88 EPHX2 (0.54) SIGMAR1AVPR1AEPHX2MAPTMAPK1
SCHEMBL3869577 0.82 EPHX2 (0.60) SIGMAR1AVPR1AEPHX2MAPTMAPK1
SCHEMBL3872069 0.82 EPHX2 (0.60) SIGMAR1AVPR1AEPHX2MAPTMAPK1
SCHEMBL3869069 0.75 CCR2 (0.69) CCR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891064-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS Laboratorios Almirall, S.A. (ES) 2008-02-27 EP claimed
WO-2006133802-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS LABORATORIOS ALMIRALL, S.A. (ES) 2006-12-21 WO claimed