SCHEMBL4673073

SCHEMBL4673073

O=C(Cc1ccsc1S(=O)(=O)c1ccc(Cl)cc1)C(=O)c1nc[nH]n1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HTT P42858 3/20 0.35
NPC1 O15118 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MAPT P10636 2/20 0.35
ADRB2 P07550 1/20 0.35
HSP90AA1 P07900 1/20 0.35
XBP1 P17861 1/20 0.35
TLR9 Q9NR96 1/20 0.35
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
AGTR1 P30556 1/20 0.34
RAB9A P51151 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
USP2 O75604 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4676736 0.90 POLB (0.37) ALDH1A1NPSR1LMNARAB9AGAA
SCHEMBL4671745 0.89 MMP1 (0.33) ALDH1A1HTTNPC1MAPTLMNA
SCHEMBL4676058 0.83 PTGER3 (0.35) ALDH1A1HTTNPC1NPSR1MAPT
SCHEMBL4671618 0.83 ALDH1A1 (0.36) ALDH1A1HTTNPC1NPSR1MAPT
SCHEMBL4676016 0.80 MAPT (0.40) ALDH1A1HTTNPC1NPSR1MAPT
SCHEMBL4672341 0.80 SMN1; SMN2 (0.35) ALDH1A1HTTMAPTSMN1; SMN2L3MBTL1
SCHEMBL4678613 0.79 ALDH1A1 (0.33) ALDH1A1HTTNPC1NPSR1MAPT
SCHEMBL4673979 0.78 NAMPT (0.33) ALDH1A1HTTMAPTHSP90AA1SMN1; SMN2
SCHEMBL4675361 0.78 NAMPT (0.33) ALDH1A1MAPTSMN1; SMN2RAB9AL3MBTL1
SCHEMBL4680019 0.78 ALDH1A1 (0.35) ALDH1A1HTTNPC1NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142872-B1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO (JP) 2008-10-15 EP disclosed
US-6620841-B1 Furan or benzofuran derivatives substituted with triazole; acquired immunodeficiency syndrome (AIDS) SHIONOGI & CO., LTD. (JP) 2003-09-16 US disclosed
EP-1142872-A1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO., LTD. (JP) 2001-10-10 EP disclosed