SCHEMBL4673283

SCHEMBL4673283

CC(=O)c1ccc(Cc2cc(C(=O)C=C(O)c3nc[nH]n3)[nH]n2)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
LMNA P02545 3/20 0.36
TSHR P16473 1/20 0.35
ALDH1A1 P00352 2/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
MAOB P27338 6/20 0.31
MAOA P21397 2/20 0.31
RXRA P19793 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4674016 0.89 MAPT (0.38) KMT2AHTTMEN1
SCHEMBL4672697 0.88 MAPT (0.38) LMNAALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL4677798 0.87 ALPL (0.34) L3MBTL1
SCHEMBL4672128 0.87 ALPL (0.34) LMNAALDH1A1L3MBTL1
SCHEMBL4677813 0.86 CYP1A2 (0.32) LMNAALDH1A1
SCHEMBL4678260 0.83 XDH (0.38) KMT2ALMNATSHRMEN1
SCHEMBL4678377 0.81 KMT2A (0.43) KMT2ALMNATSHRMEN1
SCHEMBL4673085 0.80 HCAR2 (0.42) LMNA
SCHEMBL4675403 0.80 KMT2A (0.35) KMT2ALMNATSHRALDH1A1HTT
SCHEMBL4677072 0.79 KMT2A (0.37) KMT2ALMNATSHRALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142872-B1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO (JP) 2008-10-15 EP disclosed
US-6645956-B1 1-(5-(4-fluorobenzyl)furan-2-yl)-3-hydroxy-3-(1H-1,2,4-triazol-3 -yl)-propenone; viricides; AIDS treatment SHIONOGI & CO., LTD. (JP) 2003-11-11 US disclosed
US-6620841-B1 Furan or benzofuran derivatives substituted with triazole; acquired immunodeficiency syndrome (AIDS) SHIONOGI & CO., LTD. (JP) 2003-09-16 US disclosed
EP-1142872-A1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO., LTD. (JP) 2001-10-10 EP disclosed