SCHEMBL4673785

SCHEMBL4673785

CCc1c(C(N)=O)ccnc1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.55
NOS3 P29474 1/20 0.55
PRKCI P41743 1/20 0.41
PIK3CB P42338 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
USP7 Q93009 1/20 0.39
PARP1 P09874 2/20 0.38
CDC7 O00311 2/20 0.38
NAPRT Q6XQN6 1/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
SIRT3 Q9NTG7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
EEF2K O00418 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6931488 0.86 NOS2 (0.55) NOS2NOS3PRKCIKDM4EALDH1A1
Hydrochloric Acid SCHEMBL6690850 0.85 NOS2 (0.56) NOS2NOS3PRKCIPIK3CBKDM4E
SCHEMBL14141522 0.83 NOS2 (0.51) NOS2NOS3PRKCIKDM4EALDH1A1
SCHEMBL8597943 0.82 KDM4E (0.40) NOS2NOS3PIK3CBKDM4EALDH1A1
SCHEMBL19439176 0.82 CCNC (0.41) NOS2NOS3PRKCIPIK3CBKDM4E
SCHEMBL30963968 0.81 KDM4E (0.39) NOS2NOS3PRKCIPIK3CBKDM4E
SCHEMBL5718475 0.77 CYP17A1 (0.46) NOS2NOS3PRKCIPIK3CBKDM4E
SCHEMBL1018547 0.76 PARP1 (0.42) KDM4EALDH1A1HPGDHSD17B10PARP1
SCHEMBL28917190 0.76 PRKCI (0.40) PRKCIKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5169967 0.76 NOS3 (0.52) NOS2NOS3PIK3CBKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed