SCHEMBL4674068

SCHEMBL4674068

Cc1cccc(C(=O)C(CC2CCNCC2)C2CCNCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.40
SLC6A3 Q01959 3/20 0.40
HTR2C P28335 2/20 0.40
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
CHRND Q07001 1/20 0.40
SLC6A4 P31645 2/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
GABRA4 P48169 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4672734 0.76 CPN1 (0.39) SLC6A2SLC6A3SLC6A4CHRM1
SCHEMBL4674063 0.75 SLC6A2 (0.40) SLC6A2SLC6A3HTR2CCHRNA1CHRNG
Bromide SCHEMBL11094811 0.75 MAOA (0.49) HTR2CGABRDGABRA1GABRB1GABRA5
SCHEMBL4671332 0.72 MEN1 (0.66) HTR2CGABRDGABRA1GABRB1GABRA5
SCHEMBL4676045 0.72 MEN1 (0.40) CHRNB2CHRNB4CHRNA3CHRNA4MEN1
SCHEMBL4673078 0.72 CES2 (0.42) SLC6A2SLC6A3SLC6A4CHRM1
SCHEMBL4670637 0.72 CES2 (0.39) MEN1CYP2D6KMT2ANPC1RAB9A
Bromide SCHEMBL10966281 0.71 MEN1 (0.64) HTR2CGABRDGABRA1GABRB1GABRA5
Hydrochloric Acid SCHEMBL16432330 0.71 MEN1 (0.69) HTR2CGABRDGABRA1GABRB1GABRA5
Hydrochloric Acid SCHEMBL23722031 0.70 SLC6A2 (0.45) SLC6A2SLC6A3HTR2CSLC6A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899324-A2 BENZIMIDAZOLE-CARBOXAMIDE COMPOUNDS AS 5-HT4 RECEPTOR AGONISTS Theravance, Inc. (US) 2008-03-19 EP disclosed
WO-2006127815-A2 BENZIMIDAZOLE-CARBOXAMIDE COMPOUNDS AS 5-HT4 RECEPTOR AGONISTS THERAVANCE, INC. (US) 2006-11-30 WO disclosed