Ramiprilat

Ramiprilat

SCHEMBL467411

C[C@H](N[C@@H](CCc1ccccc1)C(=O)O)C(=O)N1[C@H](C(=O)O)C[C@@H]2CCC[C@@H]21

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACE P12821 14/20 0.82
MEN1 O00255 2/20 0.82
KMT2A Q03164 2/20 0.82
CYP3A4 P08684 1/20 0.82
ALOX15 P16050 1/20 0.82
USP2 O75604 1/20 0.79
LMNA P02545 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ramiprilat SCHEMBL4634176 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL9285191 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL5490942 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL10590419 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL9438804 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL5490939 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL9594279 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL4733176 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL21990787 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15
Ramiprilat SCHEMBL9438808 1.00 ACE (0.82) ACEMEN1KMT2ACYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2085 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615449-A1 METHOD TO PREVENT AND TREAT DIABETIC RETINOPATHY BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS Weinberg, Assa (US) 2025-09-17 EP claimed
US-20250262195-A1 METHOD TO PREVENT AND TREAT DIABETIC RETINOPATHY BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS WEINBERG ASSA (US) 2025-08-21 US claimed
EP-4598526-A1 METHOD TO PREVENT AND TREAT GLAUCOMA BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS Weinberg, Assa (US) 2025-08-13 EP claimed
US-20250228831-A1 METHOD TO PREVENT AND TREAT GLAUCOMA BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS WEINBERG ASSA (US) 2025-07-17 US claimed
US-20250082608-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2025-03-13 US claimed
EP-4448096-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE Singapore Health Services Pte. Ltd. (SG) 2024-10-23 EP claimed
WO-2024102328-A1 METHOD TO PREVENT AND TREAT DIABETIC RETINOPATHY BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS WEINBERG ASSA (US) 2024-05-16 WO claimed
WO-2024076697-A1 METHOD TO PREVENT AND TREAT GLAUCOMA BY CALCIUM CHANNEL BLOCKERS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS, AND ANGIOTENSIN RECEPTOR BLOCKERS WEINBERG ASSA (US) 2024-04-11 WO claimed
EP-3474836-B1 SALBUTAMOL-CONTAINING OPHTHALMIC MEDICAMENT REKIK RAOUF (TN) 2024-01-17 EP claimed
US-20230265182-A1 USE OF IL-1 BETA BINDING ANTIBODIES TO TREAT PERIPHERAL ARTERIAL DISEASE NOVARTIS AG (CH) 2023-08-24 US claimed
WO-2001015673-A2 PHARMACEUTICAL FORMULATIONS AND USE THEREOF IN THE PREVENTION OF STROKE, DIABETES AND/OR CONGESTIVE HEART FAILURE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-08 WO claimed
US-5977159-A Medical use of an ace-inhibitor for treatment of dyspeptic symptoms ASTRA AKTIEBOLAG (SE) 1999-11-02 US claimed
CN-1207685-A Novel medical use of ACE-inhibitor for treatment of dyspeptic symptoms ASTRA AB (SE) 1999-02-10 CN claimed
EP-0835123-A1 AMINOPEPTIDASE P INHIBITORS AND USES THEREOF LOYOLA UNIVERSITY OF CHICAGO (US) 1998-04-15 EP claimed
EP-0804229-A2 COMPOSITION CONTAINING AMLODIPINE, OR A SALT OR FELODIPINE AND ANACE INHIBITOR PFIZER INC. (US) 1997-11-05 EP claimed
EP-0795327-A1 Use of Amlodipine for the treatment and prophylaxis of congestive cardiac failure of non-ischaemic origin PFIZER INC. (US) 1997-09-17 EP claimed
US-5656603-A INHIBITING BRANDYKININ DEGRADATION LOYOLA UNIVERSITY OF CHICAGO (US) 1997-08-12 US claimed
WO-1996039163-A1 AMINOPEPTIDASE P INHIBITORS AND USES THEREOF LOYOLA UNIVERSITY OF CHICAGO (US) 1996-12-12 WO claimed
WO-1996028185-A2 COMPOSITION CONTAINING AMLODIPINE, OR A SALT, OR FELODIPINE AND AN ACE INHIBITOR PFIZER INC. (US) 1996-09-19 WO claimed
EP-0391462-A1 Synergistic compositions containing ketanserin JANSSEN PHARMACEUTICA N.V. (BE) 1990-10-10 EP claimed