SCHEMBL4675591

SCHEMBL4675591

O=C(Cc1ccc(CBr)cc1)OCc1ccccc1

nearest known ligand 0.79

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.79
MAPK1 P28482 1/20 0.79
L3MBTL1 Q9Y468 1/20 0.79
PAM P19021 1/20 0.56
ENPP2 Q13822 1/20 0.52
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KMT2A Q03164 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
TSHR P16473 2/20 0.48
TRPA1 O75762 1/20 0.48
LIPE Q05469 1/20 0.48
CASP1 P29466 1/20 0.47
MGLL Q99685 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6784181 0.91 ALDH1A1 (0.96) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL361779 0.89 ALDH1A1 (1.00) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL27629121 0.87 ALDH1A1 (0.74) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL4673587 0.87 ALDH1A1 (0.69) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL2658640 0.86 ALDH1A1 (0.79) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL57331 0.86 ALDH1A1 (0.85) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL31245908 0.86 ALDH1A1 (0.85) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL27499661 0.85 ALDH1A1 (0.92) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL8117331 0.84 ALDH1A1 (0.82) ALDH1A1MAPK1L3MBTL1PAMENPP2
SCHEMBL6160393 0.83 ALDH1A1 (0.79) ALDH1A1MAPK1L3MBTL1PAMENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663936-B1 BIARYLOXYMETHYLARENE-CARBOXYLIC ACIDS HOFFMANN LA ROCHE (CH) 2008-01-09 EP disclosed
EP-1435989-A4 PTP1B INHIBITORS AND LIGANDS EINSTEIN COLL MED (US) 2006-05-03 EP disclosed
US-20040191926-A1 Ptp1b inhibitors and ligands NATIONAL INSTITUTES OF HEALTH 2004-09-30 US disclosed
EP-1435989-A1 PTP1B INHIBITORS AND LIGANDS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2004-07-14 EP disclosed
WO-2003041729-A1 PTP1B INHIBITORS AND LIGANDS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2003-05-22 WO disclosed