SCHEMBL4677367

SCHEMBL4677367

CN(CCCN1c2ccccc2CCc2ccccc21)CCC(=O)NCc1ccc(C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.53
ADORA3 P0DMS8 2/20 0.53
CHRM1 P11229 2/20 0.53
DRD2 P14416 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53
CHRM3 P20309 2/20 0.53
CNR1 P21554 2/20 0.53
SLC6A2 P23975 2/20 0.53
HTR2A P28223 2/20 0.53
HTR2C P28335 2/20 0.53
ADRA1A P35348 2/20 0.53
HRH1 P35367 2/20 0.53
DRD3 P35462 2/20 0.53
OPRK1 P41145 2/20 0.53
SLC6A3 Q01959 2/20 0.53
KCNH2 Q12809 2/20 0.53
NR1I2 O75469 1/20 0.53
ADRB2 P07550 1/20 0.53
PTGS2 P35354 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680086 0.90 SMPD1 (0.53) SLC6A4ADORA3CHRM1DRD2ADRA2B
SCHEMBL13980412 0.85 SLC6A4 (0.46) SLC6A4ADORA3CHRM1DRD2ADRA2B
SCHEMBL4733904 0.81 SLC6A4 (0.65) SLC6A4ADORA3CHRM1DRD2ADRA2B
SCHEMBL4678769 0.73 SLC6A4 (0.63) SLC6A4ADORA3CHRM1DRD2ADRA2B
Imipramine SCHEMBL20644144 0.72 SLC6A4 (0.83) SLC6A4ADORA3CHRM1DRD2ADRA2B
SCHEMBL9326845 0.72 EPHX2 (0.67) CNR1ALDH1A1LMNA
SCHEMBL7604567 0.70 SLC6A4 (0.58) SLC6A4ADORA3CHRM1DRD2ADRA2B
SCHEMBL13980489 0.69 SLC6A4 (0.73) SLC6A4ADORA3CHRM1DRD2ADRA2B
Lofepramine SCHEMBL5781415 0.69 SLC6A4 (1.00) SLC6A4ADORA3CHRM1DRD2ADRA2B
Hydrochloric Acid SCHEMBL7806943 0.69 LMNA (0.59) SLC6A4ADORA3CHRM1DRD2ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216994-B1 Tricyclic antidepressant derivatives and immunoassay ROCHE DIAGNOSTICS GMBH (DE) 2008-12-31 EP disclosed
EP-1216994-B1 Tricyclic antidepressant derivatives and immunoassay ROCHE DIAGNOSTICS GMBH (DE) 2008-12-31 EP disclosed
EP-1216994-A2 Tricyclic antidepressant derivatives and immunoassay Roche Diagnostics GmbH (DE) 2002-06-26 EP disclosed
US-6368814-B1 TRICYCLIC ANTIDEPRESSANTS AND METABOLITES THEREOF ROCHE DIAGNOSTICS CORPORATION 2002-04-09 US disclosed