SCHEMBL4679446

SCHEMBL4679446

C[C@H](C(=O)O)c1ccc2ccccc2c1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.69
AKR1C3 P42330 13/20 0.67
AKR1C2 P52895 13/20 0.67
PTGS2 P35354 4/20 0.67
PTGS1 P23219 3/20 0.67
CDC42 P60953 1/20 0.67
RAC1 P63000 1/20 0.67
CYP1A2 P05177 1/20 0.67
TSHR P16473 1/20 0.67
SLC22A6 Q4U2R8 1/20 0.67
UGT2B7 P16662 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12431128 1.00 AKR1B1 (0.69) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL30717241 1.00 AKR1B1 (0.69) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL10025981 1.00 AKR1B1 (0.69) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL1217681 1.00 AKR1B1 (0.69) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
Hydrochloric Acid SCHEMBL27401798 0.98 AKR1B1 (0.67) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL503391 0.93 AKR1B1 (0.61) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL11470486 0.90 AKR1C3 (0.69) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
Naproxen SCHEMBL23753934 0.89 AKR1C3 (0.88) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
Ammonia Solution, Strong SCHEMBL11721423 0.89 AKR1C3 (0.67) AKR1B1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL15695558 0.89 UGT2B7 (0.60) AKR1B1AKR1C3AKR1C2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024010529-A1 PRODUCTION OF ENANTIOPURE ALCOHOLS, AMINES AND ACIDS FROM RACEMIC EPOXIDES BY CASCADE BIOTRANSFORMATION INVOLVING EPOXIDE ISOMERIZATION AND DYNAMIC KINETIC RESOLUTION NATIONAL UNIVERSITY OF SINGAPORE (SG) 2024-01-11 WO disclosed
WO-2013028132-A9 CHIRAL PHOSPHINES FOR PALLADIUM-CATALYZED ASYMMETRIC ALPHA-ARYLATION OF ESTER ENOLATES TO PRODUCE TERTIARY STEREOCENTERS IN HIGH ENANTIOSELECTIVITY NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2013-08-22 WO disclosed
US-8268865-B2 Quaternary alkyl ammonium bacterial efflux pump inhibitors and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2012-09-18 US disclosed
US-20120165276-A1 QUATERNARY ALKYL AMMONIUM BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF MPEX PHARMACEUTICALS, INC. (US) 2012-06-28 US disclosed
US-20120077976-A1 CAMPHOR-DERIVED COMPOUNDS, METHOD FOR MANUFACTURING THE SAME, AND APPLICATION THEREOF NATIONAL TSING HUA UNIVERSITY (TW) 2012-03-29 US disclosed
US-20120077976-A1 CAMPHOR-DERIVED COMPOUNDS, METHOD FOR MANUFACTURING THE SAME, AND APPLICATION THEREOF NATIONAL TSING HUA UNIVERSITY (TW) 2012-03-29 US disclosed
EP-1045836-B1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMA (US) 2008-03-05 EP disclosed
EP-1045836-B1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMA (US) 2008-03-05 EP disclosed
CN-1128874-C Rhodococcus sp.D12 and its culture method and application SHANGHAI INST ORGANIC CHEM (CN) 2003-11-26 CN disclosed
US-6284768-B1 Src family SH2 domain inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2001-09-04 US disclosed
US-6268365-B1 Src family SH2 domain inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2001-07-31 US disclosed
CN-1291648-A Rhodococcus sp.D12 and its culture method and application SHANGHAI INST ORGANIC CHEM (CN) 2001-04-18 CN disclosed
EP-1045836-A1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2000-10-25 EP disclosed
US-6054470-A Src family SH2 domain inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-04-25 US disclosed
WO-1999031066-A1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1999-06-24 WO disclosed
EP-0314759-A4 ASYMMETRIC HYDROFORMYLATIONS OF PROCHIRAL OLEFINS TO CHIRAL ALDEHYDES IN HIGH ENANTIOMERIC EXCESS. UNIV COLORADO STATE RES FOUND (US) 1990-01-29 EP disclosed
EP-0314759-A1 ASYMMETRIC HYDROFORMYLATIONS OF PROCHIRAL OLEFINS TO CHIRAL ALDEHYDES IN HIGH ENANTIOMERIC EXCESS COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1989-05-10 EP disclosed
WO-1988008835-A1 ASYMMETRIC HYDROFORMYLATIONS OF PROCHIRAL OLEFINS TO CHIRAL ALDEHYDES IN HIGH ENANTIOMERIC EXCESS COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1988-11-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077976-A1 CAMPHOR-DERIVED COMPOUNDS, METHOD FOR MANUFACTURING THE SAME, AND APPLICATION THEREOF PDE10A, PDE6H, PRKAR2A AKR1B1 218/4885AKR1C3 77/4885AKR1C2 169/4885
US-20120165276-A1 QUATERNARY ALKYL AMMONIUM BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF ABCB11, ABCC1, SLC47A1 AKR1B1 2198/4885AKR1C3 3170/4885AKR1C2 2657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.